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Scopus Author ID: 6506811439

Communications and Full papers

44 - Total Synthesis of a Pancratistatin/Shikimic Acid Hybrid Analogue Azubuike D, Di Iulio GA, Caggiano L  Eur.JOC, 2024, e202301247.

42 - Exploring Convergent Two-Step Synthetic Approaches to the Pancratistatin Framework Di Iulio GA, Mahon MF, Caggiano L ChemistrySelect, 20227, e202202703.

40 - Stuart Warren (24 Dec 1938–22 Mar 2020) Aggarwal VK, Armstrong SK, Caggiano L, Chibale K, Clayden J, Coldham I, Greeves N, Hartley RC, Knight JG, Kuhnert N, Mitchell HJ, Nelson A, O'Brien P, Thomas SP and Wyatt P. Org. Biomol. Chem., 2020, 18, 7236-7237.

39 - NADPH oxidase 1 is a novel pharmacological target for the development of an antiplatelet drug without bleeding side effects. Vara D, Tarafdar A, Celikag M, Patinha D, Gulacsy CE, Hounslea E, Warren Z, Ferreira B, Koeners MP, Caggiano L and Pula G. The FASEB Journal, 2020, 34(10), 13959-13977. Open Access

38 - Sidechain diversification of grandifloracin allows identification of analogues with enhanced anti-austerity activity against human PANC-1 pancreatic cancer cells. Alexander BE, Sun S, Palframan MJ, Kociok-Köhn G, Caggiano L, Awale S and Lewis SE ChemMedChem, 2020, 14, 125-135 Open Access

37 - Novel NADPH oxidase 1-selective inhibitors impair collagen-dependent platelet activation and thrombus formation in vitro and ferric chloride-induced carotid occlusion in vivo with negligible effects on thrombin responses and bleeding time. Vara D, Tarafdar A, Caggiano L and Pula G Free Radical Biology and Medicine, 2019, 139, S55

35 - The Enone Motif of (+)-Grandifloracin is Not Essential for "Anti-Austerity" Anti-proliferative Activity. Khan MA, Wood PJ, Lamb-Guhren NM, Caggiano L, Kociok-Köhn G, Tosh D and Lewis SE Bioorg. Med. Chem. Lett., 2014, 24, 2815-2819 Open Access

34 - Design, synthesis and antiproliferative activity of indole analogues of indanocine. Tunbridge GA, Oram J and Caggiano L MedChemComm, 2013, 4, 1452-1456 Open Access

Highlighted by the Editors of MedChemComm as one of the most accessed articles of 2013!!!

33 - Multicellular aggregation of maltol-modified cells triggered by Fe(III) ions. Ciupa A, De Bank PA and Caggiano L ChemCommun., 201349, 10148-10150 Open Access

32 - Synthesis and antiproliferative activity of some 3-(pyrid-2-yl)-pyrazolines. Ciupa A, De Bank PA, Mahon MF, Wood PJ and Caggiano L MedChemComm, 2013, 4, 956 - 961 Open Access

Second most accessed article in the 2nd quarter of 2013! A list of the top ten is provided. Also highlighted by the Editors of MedChemComm as one of the most accessed articles of 2013!!!

30 - Mild and Efficient Capture and Functionalisation of CO2 using Silver(I) Oxide and Application to 13C-labelled Dialkyl Carbonates. Tunbridge GA, Baruchello R and Caggiano L RSC Advances, 2013, 3, 4613 - 4621

28 - Simple pyrazoline and pyrazole "turn on" fluorescent sensors selective for Cd2+ and Zn2+ in MeCN. Ciupa A, Mahon MF, De Bank PA and Caggiano L Org. Biomol. Chem., 2012, 10, 8753-8757

27 - Design, synthesis and antiproliferative activity of urocanic-chalcone hybrid derivatives. Ciupa A, Griffiths NJ, Light SK, Wood PJ and Caggiano L MedChemComm 2011, 2, 1011-1015

Listed in the "Top ten accessed articles in September 2011"

26 - Bi(OTf)3-catalysed prenylation of electron-rich aryl ethers and phenols with isoprene: a direct route to prenylated derivatives. Judd KE and Caggiano L Org. Biomol. Chem., 2011, 9, 5201-5210

24 - Application of Negishi Cross-Coupling to the Synthesis of the Cyclic Tripeptides OF-4949-III and K-13. Nolasco L; Perez-Gonzalez M; Caggiano L and Jackson RFW. J. Org. Chem., 2009, 74, 8280-8289

23 - Efficient Synthesis of Tetrahydro-b-carbolin-1-one and Dihydroisoquinolin-1-one Derivatives as Versatile Intermediates. Judd KE; Mahon MF and Caggiano L. Synthesis, 2009, 16, 2809-2817

22 - Enantioselective oxidation of an alkyl aryl sulfide. Drago C; Walker EJ; Caggiano L and Jackson RFW. Org. Synth., 2009, 86, 121-129

21 - Ionization of the Zinc/Iodine Bond of Alkylzinc Iodides in Dimethylformamide from Theory and Experiment. Caggiano L; Jackson RFW; Meijer AJHM, Pickup BT and Wilkinson KA. Chem. Eur. J., 2008, 14, 8798-8802

20 - alpha-Fluorination of beta-keto sulfones by Selectfluor™. Loghmani-khouzani H; Poorheravi MR; Sadeghi MMM; Caggiano L and Jackson RFW. Tetrahedron, 2008, 64, 7419-7425

19 - Synthesis of beta-2-homophenylalanine derivatives by Negishi cross-coupling reactions. Bartrum HE; Adams H; Caggiano L and Jackson RFW. Tetrahedron, 2008, 64, 3701-3712

18 - Negishi cross-coupling reactions of alpha-amino acid-derived organozinc reagents with aromatic bromides. Oswald CL, Carrillo-Márquez T, Caggiano L and Jackson RFW. Tetrahedron, 2008, 64, 681-687

17 - Stereoselective synthesis of 2,3-difunctionalised thioesters using nucleophilic epoxidation of 1-arylthio-1-nitroalkenes. Evans LA, Adams H, Barber CG, Caggiano L and Jackson RFW. Org. Biomol. Chem., 2007, 5, 3156-3163

16 - Oxidative Kinetic Resolution of Alkyl Aryl Sulfoxides. Mohammadpoor-Baltork I, Hill M, Caggiano L and Jackson RFW. Synlett, 2006, 20, 3540–3544

15 - Synthesis of orthogonally protected biaryl amino acid derivatives. Moreno E, Nolasco LA, Caggiano L and Jackson RFW. Org. Biomol. Chem., 2006, 4, 3639–3647

14 - Effective Asymmetric Oxidation of Enones and Alkyl Aryl Sulfides. Hinch M, Jacques O, Drago C, Caggiano L, Jackson RFW, Dexter C, Anson MS and Macdonald SJF. Journal of Molecular Catalysis A: Chemical, 2006, 251 (1-2), 123-128

13 - A Formal Total Synthesis of Eleutherobin Using the Ring-Closing-Metathesis Reaction of a Densely Functionalized Diene as the Key-Step: Investigation of the Unusual Kinetically-Controlled RCM Stereochemistry. Castoldi D, Caggiano L, Panigada L, Sharon O, Costa A M and Gennari C. Chem. Eur. J. 2006, 12, 51-62

Graphical abstract

12 - Vanadium-Catalysed Sulfur Oxidation/Kinetic Resolution Process for the Synthesis of Enantiomerically Pure Alkyl Aryl Sulfoxides. Drago C, Caggiano L and Jackson RFW. Angew. Chem. Int. Ed., 2005, 44, 7221-7223

10 - New routes to ß–cycloalkane derivatives using serine-derived organozinc reagents. Carrillo-Marquez T, Caggiano L, Jackson RFW, Graboswka U, Rae A, Tozer MJ. Org. Biomol. Chem. 2005, 3, 4117-4123

9 - Synthesis of novel, simplified, C-7 substituted eleutheside analogues with potent microtubule-stabilizing activity. Castoldi D, Caggiano L, Bayón P, Costa A M, Cappella P, Sharon O and Gennari C. Tetrahedron, 2005, 61, 2123-2139

8 - A formal total synthesis of eleutherobin through an unprecedented kinetically controlled ring-closing-metathesis reaction of a densely functionalized diene. Castoldi D, Caggiano L, Panigada L, Sharon O, Costa A M and Gennari C. Angew. Chem. Int. Ed., 2005, 44, 588-591

7 - Effects of allylic and homoallylic substituents on the ring closing metathesis reaction used to synthesise simplified eleuthesides. Caggiano L, Castoldi D, Beumer R, Bayón P, Telser J and Gennari C. Tet. Lett., 2003, 44, 7913-7919

6 - Novel silica catalyzed stereoselective cyclic carbamate and carbonate rearrangements. Caggiano L, Davies J, Fox DJ, Moody DM, Warren S. Chem. Commun., 2003, 14, 1650-1652

5 - Stereoselective substituted pyrrolidine and cyclic ether synthesis by PhS migration. Caggiano L, Davies J, Fox DJ, Moody DM, Warren S. Chem. Commun., 2003, 14, 1648-1650

4 - Silica gel catalyzed generation of episulfonium ions: a mild method for the synthesis of heterocycles. Caggiano L, Fox DJ, Warren S. Chem. Commun., 2002, 23, 2528-2529

3 - Asymmetric synthesis of tetrahydropyrans with competitive [1,2]-phenylsulfanyl (PhS) migrations. Caggiano L, Fox DJ, House D, Jones ZA, Kerr F, Warren S. JCS-Perkin Trans. 1., 2002, 23, 2646-2651

2 - Asymmetric synthesis of tetrahydrofurans by competitive [1,2]-phenylsulfanyl (PhS) migrations under thermodynamic control. Caggiano L, Fox DJ, House D, Jones ZA, Kerr F, Warren S. JCS-Perkin Trans. 1., 2002, 23, 2634-2645

Review Article

11 - Organozinc halides in organic synthesis. Rilatt I, Caggiano L, Jackson RFW. Synlett 2005, 18, 2701-2719

PhD Theses

1 - Silica Gel Induced Episulfonium Ion Formation and Capture with Internal Nucleophiles. Caggiano, L. 2002.
Supervisor Dr Stuart Warren.

25 - Synthesis and Evaluation of Narciclasine Analgoues. Judd, K. 2011.
Supervisor Dr Lorenzo Caggiano.

29 - Efficient Synthesis of Biologically Active Small Molecules. Tunbridge, G. 2012.
Supervisor Dr Lorenzo Caggiano.

31 - Chalcone Derivatives in Cancer Research and Tissue Engineering. Ciupa, A. 2013.
Supervisor Dr Lorenzo Caggiano.

36 - Design, Synthesis and Biological Activity of Narciclasine Analogues. Griffiths, N. 2015.
Supervisor Dr Lorenzo Caggiano.

41 - Design and Synthesis of Novel Narciclasine/Pancratistatin Analogues as Potential Brain-Tumour Agents. Azubuike, D. 2021.
Supervisor Dr Lorenzo Caggiano.

43 - Investigation of a Diels-Alder Approach to Novel Narciclasine Derivatives . Xu, Haoran. 2023.
Supervisor Dr Lorenzo Caggiano.

Book Reviews

An introduction to Medicinal Chemistry, Fifth Edition by Graham L. Patrick.
Caggiano L. Chemistry World, 2013

Silicon-mediated Transformations of Functional Groups by Helmut Vorbrueggen.
Caggiano L. Applied Organometallic Chemistry, 2005, 19, 699


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